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Found 130 with Last Name = 'timmers' and Initial = 'cm'
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376888(CHEMBL415279)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376892(CHEMBL406958)
Affinity DataKi:  170nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376889(CHEMBL260647)
Affinity DataKi:  260nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376893(CHEMBL262334)
Affinity DataKi:  380nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376878(CHEMBL436906)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376877(CHEMBL259878)
Affinity DataKi:  480nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376883(CHEMBL404611)
Affinity DataKi:  500nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376873(CHEMBL438168)
Affinity DataKi:  510nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376896(CHEMBL262599)
Affinity DataKi:  530nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376890(CHEMBL261649)
Affinity DataKi:  580nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376895(CHEMBL406960)
Affinity DataKi:  600nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376875(CHEMBL260812)
Affinity DataKi:  620nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376899(CHEMBL260318)
Affinity DataKi:  700nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376876(CHEMBL408760)
Affinity DataKi:  720nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376874(CHEMBL260750)
Affinity DataKi:  740nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376891(CHEMBL439076)
Affinity DataKi:  770nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376880(CHEMBL436862)
Affinity DataKi:  820nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376885(CHEMBL262335)
Affinity DataKi:  840nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376884(CHEMBL429690)
Affinity DataKi:  850nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376897(CHEMBL406084)
Affinity DataKi:  930nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376879(CHEMBL266172)
Affinity DataKi:  930nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376900(CHEMBL258970)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376898(CHEMBL408759)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376894(CHEMBL259220)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376881(CHEMBL406713)
Affinity DataKi:  2.20E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376887(CHEMBL436878)
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376886(CHEMBL436697)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50376882(CHEMBL437260)
Affinity DataKi:  5.30E+3nMAssay Description:Displacement of [125I]triptorelin from human GnRHR expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410306(CHEMBL436481)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410307(CHEMBL360981)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410303(CHEMBL361847)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410309(CHEMBL365545)
Affinity DataIC50:  9nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of maximum response evoked by cAMP on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyrotropin receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM60862(BDBM189328 | US9174940, 32)
Affinity DataIC50:  12nMAssay Description:Antagonist activity of three test compounds against human TSI at the human TSH receptor was tested in Chinese Hamster Ovary (CHO) cells (cultured 16 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410304(CHEMBL195469)
Affinity DataIC50:  25nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410302(CHEMBL361167)
Affinity DataIC50:  27nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50162936(Biphenyl-4-carboxylic acid (1-acetyl-2,2,4-trimeth...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410308(CHEMBL192868)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410298(CHEMBL178980)
Affinity DataIC50:  31nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50335479((R)-N-(1-acetyl-2,2,4-trimethyl-4-(4-(prop-2-ynylo...)
Affinity DataIC50:  39nMAssay Description:Agonist activity at human FSHR receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyrotropin receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM189329((+)-(1-Acetyl-4-methyl-4-phenyl-1,2,3,4-tetrahydro...)
Affinity DataIC50:  47nMAssay Description:Antagonist activity of three test compounds against human TSI at the human TSH receptor was tested in Chinese Hamster Ovary (CHO) cells (cultured 16 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetThyrotropin subunit beta(Bos taurus (Bovine))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM60862(BDBM189328 | US9174940, 32)
Affinity DataIC50:  48nMAssay Description:Antagonist activity of three test compounds against human TSI at the human TSH receptor was tested in Chinese Hamster Ovary (CHO) cells (cultured 16 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410294(CHEMBL195347)
Affinity DataIC50:  50nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410292(CHEMBL192334)
Affinity DataIC50:  54nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50115998(3-[(Benzyl-methyl-amino)-methyl]-8-(2,6-difluoro-b...)
Affinity DataIC50:  71nMAssay Description:Antagonist activity at human GnRHR expressed in CHO cells after 30 mins by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Research And Development

Curated by ChEMBL
LigandPNGBDBM50410300(CHEMBL179505)
Affinity DataIC50:  76nMAssay Description:In vitro inhibition of maximum response on CHO-K1 cells expressing human Follicle stimulating hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyrotropin receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM189327(Hexanoic acid (Compound A) | US9174940, Compound A)
Affinity DataIC50:  88nMAssay Description:Antagonist activity of three test compounds against human TSI at the human TSH receptor was tested in Chinese Hamster Ovary (CHO) cells (cultured 16 ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetThyrotropin receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM60860(US9174940, 31)
Affinity DataIC50: <100nMAssay Description:Antagonist activity of three test compounds against human TSI at the human TSH receptor was tested in Chinese Hamster Ovary (CHO) cells (cultured 16 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetThyrotropin receptor(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM60862(BDBM189328 | US9174940, 32)
Affinity DataIC50: <100nMAssay Description:Antagonist activity of three test compounds against human TSI at the human TSH receptor was tested in Chinese Hamster Ovary (CHO) cells (cultured 16 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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