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Found 122 with Last Name = 'toney' and Initial = 'jh'
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042574(5-Butyl-2-(2,5-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataKi:  8.00E+4nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042531(5-Butyl-2-(2,3-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataKi:  1.70E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042561(5-Butyl-2-(2-chloro-phenyl)-4-[2'-(1H-tetrazol-5-y...)
Affinity DataKi:  2.50E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042579(5-Butyl-2-phenyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  2.50E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042542(5-Butyl-2-(2,3-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataKi:  3.10E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042559(5-Butyl-2-(2-chloro-phenyl)-4-[2'-(1H-tetrazol-5-y...)
Affinity DataKi:  3.50E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042578(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  3.80E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042577(5-Butyl-2-(2,5-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataKi:  3.80E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042564(5-Butyl-2-(4-chloro-phenyl)-4-[2'-(1H-tetrazol-5-y...)
Affinity DataKi:  3.80E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042543(5-Butyl-2-(2,4-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataKi:  4.00E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042558(2-Biphenyl-2-yl-5-butyl-4-[2'-(1H-tetrazol-5-yl)-b...)
Affinity DataKi:  4.20E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042535(5-Butyl-2-(3-chloro-phenyl)-4-[2'-(1H-tetrazol-5-y...)
Affinity DataKi:  4.25E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042556(5-Butyl-2-(4-chloro-phenyl)-4-[2'-(1H-tetrazol-5-y...)
Affinity DataKi:  4.30E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042528(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  4.50E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042548(5-Butyl-2-(3-chloro-phenyl)-4-[2'-(1H-tetrazol-5-y...)
Affinity DataKi:  4.50E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042569(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  4.70E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042568(5-Butyl-2-(2,4-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataKi:  4.80E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042565(5-Butyl-2-(2,6-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataKi:  5.00E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042555(5-Butyl-2-phenyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  5.90E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042544(5-Butyl-2-(2-nitro-phenyl)-4-[2'-(1H-tetrazol-5-yl...)
Affinity DataKi:  6.40E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(GUINEA PIG)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042576(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  8.00E+5nMAssay Description:In vitro apparent inhibition constant of porcine renal Dehydropeptidase-1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36643(L-161,189)
Affinity DataIC50:  300nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36644(L-159,906)
Affinity DataIC50:  400nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36639(L-158-817)
Affinity DataIC50:  1.80E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36640(CHEMBL26514 | L-159,061)
Affinity DataIC50:  1.90E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36638(L-158-678)
Affinity DataIC50:  3.50E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36636(L-809-559)
Affinity DataIC50:  4.00E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36642(L-809,370)
Affinity DataIC50:  6.00E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36645(CHEMBL291582 | L-707,581)
Affinity DataIC50:  7.00E+3nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Escherichia coli)
Merck Research Laboratorie

Curated by ChEMBL
LigandPNGBDBM50081042((R)-3-Dibenzofuran-2-yl-2-mercapto-propionic acid ...)
Affinity DataIC50:  9.90E+3nMAssay Description:Inhibitory activity against CCRA (B. fragilis) metallo-beta-lactamaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042557(5-Butyl-2-(2-nitro-phenyl)-4-[2'-(1H-tetrazol-5-yl...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042540(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042559(5-Butyl-2-(2-chloro-phenyl)-4-[2'-(1H-tetrazol-5-y...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042576(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042542(5-Butyl-2-(2,3-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042578(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36641(L-809,339)
Affinity DataIC50:  4.20E+4nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Bacteroides fragilis)
Merck Research Laboratories

LigandPNGBDBM36637(L-809-558)
Affinity DataIC50:  4.20E+4nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using metallo-beta-lactamase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042577(5-Butyl-2-(2,5-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042574(5-Butyl-2-(2,5-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Pseudomonas aeruginosa mediated by the plasmid-borne IMP-1 enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042558(2-Biphenyl-2-yl-5-butyl-4-[2'-(1H-tetrazol-5-yl)-b...)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Pseudomonas aeruginosa mediated by the plasmid-borne IMP-1 enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042568(5-Butyl-2-(2,4-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Pseudomonas aeruginosa mediated by the plasmid-borne IMP-1 enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042564(5-Butyl-2-(4-chloro-phenyl)-4-[2'-(1H-tetrazol-5-y...)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Pseudomonas aeruginosa mediated by the plasmid-borne IMP-1 enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042532(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-lactamase(Pseudomonas aeruginosa)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042548(5-Butyl-2-(3-chloro-phenyl)-4-[2'-(1H-tetrazol-5-y...)
Affinity DataIC50:  7.60E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Pseudomonas aeruginosa mediated by the plasmid-borne IMP-1 enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042569(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042528(5-Butyl-4-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetallo-beta-lactamase type 2(Bacteroides fragilis)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50042543(5-Butyl-2-(2,4-dichloro-phenyl)-4-[2'-(1H-tetrazol...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of metallo-beta-lactamase (MBL) from Bacteroides fragilis.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36639(L-158-817)
Affinity DataIC50: >1.00E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidase 1(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM36640(CHEMBL26514 | L-159,061)
Affinity DataIC50: >1.00E+5nMpH: 7.0 T: 2°CAssay Description:Enzyme inhibition assay by biphenyl tetrazoles (BPTS)using dehydropeptidase 1 (DPH-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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