Affinity DataKi: 0.100nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 0.620nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 3 receptor was evaluatedMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 0.794nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 3 receptor was evaluatedMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Universidade Estadual De Feira De Santana
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity towards 5-HT4 receptor in striatum membranes of guinea-pig brain was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 11.2nMAssay Description:Binding affinity towards 5-HT3 receptor in rat was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity to bovine thrombin assessed as inhibition constant using tosyl-Gly-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 13.8nMAssay Description:Binding affinity towards 5-HT3 receptor in rat was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity towards 5-HT3 receptor in rat was evaluatedMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity to bovine thrombin assessed as inhibition constant using tosyl-Gly-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 58nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataKi: 59nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Binding affinity to bovine thrombin assessed as inhibition constant using tosyl-Gly-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor in striatum membranes of guinea-pig brain was evaluatedMore data for this Ligand-Target Pair