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Found 659 with Last Name = 'villa' and Initial = 'f'
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592222(CHEMBL5180135)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50103072(1-Benzyl-2-piperazin-1-yl-1H-benzoimidazole | CHEM...)
Affinity DataKi:  0.620nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 3 receptor was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592224(CHEMBL5193920)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50258672(CHEMBL513681 | [4-(2,3,4,5-Tetrahydro-1,3-dimethyl...)
Affinity DataKi:  0.794nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592225(CHEMBL5207279)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592222(CHEMBL5180135)
Affinity DataKi:  1nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50282641(CHEMBL4160732)
Affinity DataKi:  1nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50282638(CHEMBL4175851)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards rat 5-hydroxytryptamine 3 receptor was evaluatedMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50282631(CHEMBL4175454)
Affinity DataKi:  1.80nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592212(CHEMBL5182038)
Affinity DataKi:  2nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592212(CHEMBL5182038)
Affinity DataKi:  3nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592211(CHEMBL5204462)
Affinity DataKi:  3nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592232(CHEMBL5196327)
Affinity DataKi:  3nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592231(CHEMBL5177749)
Affinity DataKi:  4nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592223(CHEMBL5204622)
Affinity DataKi:  4nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592232(CHEMBL5196327)
Affinity DataKi:  4nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592231(CHEMBL5177749)
Affinity DataKi:  5nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universidade Estadual De Feira De Santana

Curated by ChEMBL
LigandPNGBDBM50233089(8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at Adenosine receptor subtype 2B in human RBC assessed as change in erythrocyte morphology incubated for 3 hrs with occasional ge...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592228(CHEMBL5204191)
Affinity DataKi:  7nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592211(CHEMBL5204462)
Affinity DataKi:  8nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592226(CHEMBL5198091)
Affinity DataKi:  9nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592224(CHEMBL5193920)
Affinity DataKi:  9nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592213(CHEMBL5182510)
Affinity DataKi:  10nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592223(CHEMBL5204622)
Affinity DataKi:  10nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592219(CHEMBL5195140)
Affinity DataKi:  11nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108391(4-Amino-5-chloro-2-methoxy-benzoic acid 2-methyl-2...)
Affinity DataKi:  11nMAssay Description:Binding affinity towards 5-HT4 receptor in striatum membranes of guinea-pig brain was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108391(4-Amino-5-chloro-2-methoxy-benzoic acid 2-methyl-2...)
Affinity DataKi:  11.2nMAssay Description:Binding affinity towards 5-HT3 receptor in rat was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592215(CHEMBL5205860)
Affinity DataKi:  12nMAssay Description:Binding affinity to bovine thrombin assessed as inhibition constant using tosyl-Gly-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592214(CHEMBL5208647)
Affinity DataKi:  13nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108388(4-Amino-5-chloro-2-methoxy-benzoic acid 2-methyl-2...)
Affinity DataKi:  13.8nMAssay Description:Binding affinity towards 5-HT3 receptor in rat was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rattus norvegicus)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108388(4-Amino-5-chloro-2-methoxy-benzoic acid 2-methyl-2...)
Affinity DataKi:  14nMAssay Description:Binding affinity towards 5-HT3 receptor in rat was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592221(CHEMBL5206845)
Affinity DataKi:  15nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592215(CHEMBL5205860)
Affinity DataKi:  17nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592210(CHEMBL5201137)
Affinity DataKi:  23nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592229(CHEMBL5188015)
Affinity DataKi:  24nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592210(CHEMBL5201137)
Affinity DataKi:  26nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592228(CHEMBL5204191)
Affinity DataKi:  28nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592218(CHEMBL5195073)
Affinity DataKi:  33nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592213(CHEMBL5182510)
Affinity DataKi:  38nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProthrombin(Bos taurus (Bovine))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592216(CHEMBL5180406)
Affinity DataKi:  42nMAssay Description:Binding affinity to bovine thrombin assessed as inhibition constant using tosyl-Gly-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592217(CHEMBL5171112)
Affinity DataKi:  43nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592220(CHEMBL5183649)
Affinity DataKi:  50nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592220(CHEMBL5183649)
Affinity DataKi:  51nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592215(CHEMBL5205860)
Affinity DataKi:  52nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592230(CHEMBL5174823)
Affinity DataKi:  58nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592218(CHEMBL5195073)
Affinity DataKi:  59nMAssay Description:Binding affinity to N-terminal MRGS(His)6GSDDDDK-tagged Matriptase (unknown origin) expressed in Escherichia coli assessed as inhibition constant usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592219(CHEMBL5195140)
Affinity DataKi:  60nMAssay Description:Binding affinity to FXa (unknown origin) using Mes-DArg-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProthrombin(Bos taurus (Bovine))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50592214(CHEMBL5208647)
Affinity DataKi:  73nMAssay Description:Binding affinity to bovine thrombin assessed as inhibition constant using tosyl-Gly-Pro-Arg-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Universidad De Alcal£

Curated by ChEMBL
LigandPNGBDBM50108391(4-Amino-5-chloro-2-methoxy-benzoic acid 2-methyl-2...)
Affinity DataKi:  83nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor in striatum membranes of guinea-pig brain was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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