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Found 816 with Last Name = 'welsh' and Initial = 'wj'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50404011(CHEMBL36900)
Affinity DataKi:  0.0100nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50473991(CHEMBL416783)
Affinity DataKi:  0.0200nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM164((4R,5R,6R)-4-benzyl-5-hydroxy-1,3-bis(1H-indazol-5...)
Affinity DataKi:  0.0200nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50404007(CHEMBL116517)
Affinity DataKi:  0.0200nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50065089((4R,5R,6R)-Tetrahydro-1,3-bis[(3-benzamide oxime)-...)
Affinity DataKi:  0.0200nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50404010(CHEMBL324293)
Affinity DataKi:  0.0302nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50473996(CHEMBL291004)
Affinity DataKi:  0.0302nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50473992(CHEMBL416612)
Affinity DataKi:  0.0603nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50404006(CHEMBL366576)
Affinity DataKi:  0.0603nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1149((4R,5R,6R)-Tetrahydro-1-(3-aminophenyl-methyl)-3-[...)
Affinity DataKi:  0.0603nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1144((4R,5R,6R)-1-[(3-aminophenyl)methyl]-4-benzyl-5-hy...)
Affinity DataKi:  0.0794nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50404005(CHEMBL113884)
Affinity DataKi:  0.0794nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1080((4R,5R,6R)-Tetrahydro-1,3-bis[(3-benzamido)methyl]...)
Affinity DataKi:  0.0891nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1148((4R,5R,6R)-1-[(3-amino-1H-indazol-5-yl)methyl]-3-[...)
Affinity DataKi:  0.100nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1145((4R,5R,6R)-1-[(3-aminophenyl)methyl]-6-benzyl-5-hy...)
Affinity DataKi:  0.100nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1109((4R,5R,6R)-4-benzyl-5-hydroxy-1,3-bis[(3-methyl-1H...)
Affinity DataKi:  0.100nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1107((4R,5R,6R)-4-benzyl-5-hydroxy-6-(2-phenylethyl)-1,...)
Affinity DataKi:  0.100nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Saint Louis University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50067497((2S,4S,4aS,6R,8aR)-4-[4-(1,1-Dimethyl-heptyl)-2-hy...)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]CP-55,940 binding to Cannabinoid receptor 1 in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1146((4R,5R,6R)-1-[(3-aminophenyl)methyl]-6-benzyl-5-hy...)
Affinity DataKi:  0.129nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1102((4R,5R,6R)-Tetrahydro-1,3-bis[(3-carboxamidophenyl...)
Affinity DataKi:  0.151nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  0.220nMAssay Description:Binding affinity against Opioid receptor delta 1 from rat brain membranes using [3H]DADLEChecked by AuthorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Saint Louis University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3(1,1-dimethylheptyl)-9-hydroxymethyl)-...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]CP-55,940 binding to Cannabinoid receptor 1 in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50473993(CHEMBL286159)
Affinity DataKi:  0.240nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1090((4R,5R,6R)-1,3-bis[(3-amino-4-fluorophenyl)methyl]...)
Affinity DataKi:  0.251nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50473997(CHEMBL36581)
Affinity DataKi:  0.282nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1089((4R,5R,6R)-4-benzyl-5-hydroxy-1,3-bis[(3-hydroxyph...)
Affinity DataKi:  0.302nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1101((4R,5R,6R)-Tetrahydro-1,3-bis[(3-carboxamidophenyl...)
Affinity DataKi:  0.309nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002109(CHEMBL370735)
Affinity DataKi:  0.340nMAssay Description:Binding affinity against Opioid receptor mu 1 from rat brain membranes using [3H]DAMGOChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50473995(CHEMBL36437)
Affinity DataKi:  0.380nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002106(CHEMBL370966)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against Opioid receptor mu 1 from rat brain membranes using [3H]DAMGOChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1111((4R,5R,6R)-1,3-bis[(3-amino-1,2-benzoxazol-5-yl)me...)
Affinity DataKi:  0.407nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1079((4R,5R,6R)-4-benzyl-5-hydroxy-1,3-bis({[3-(hydroxy...)
Affinity DataKi:  0.490nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
The State University Of New Jersey

Curated by ChEMBL
LigandPNGBDBM50566013(CHEMBL4800218)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain membranes incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50473990(CHEMBL431321)
Affinity DataKi:  0.646nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002059(CHEMBL606795)
Affinity DataKi:  0.710nMAssay Description:Binding affinity against Opioid receptor delta 1 from rat brain membranes using [3H]DADLEChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002069(CHEMBL611398)
Affinity DataKi:  0.710nMAssay Description:Binding affinity against Opioid receptor delta 1 from rat brain membranes using [3H]DADLEChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002041(CHEMBL195784)
Affinity DataKi:  0.780nMAssay Description:Binding affinity against Opioid receptor delta 1 from rat brain membranes using [3H]DADLEChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002081(CHEMBL610798)
Affinity DataKi:  0.790nMAssay Description:Binding affinity against Opioid receptor delta 1 from rat brain membranes using [3H]DADLEChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002111(CHEMBL371845)
Affinity DataKi:  0.830nMAssay Description:Binding affinity against Opioid receptor mu 1 from rat brain membranes using [3H]DAMGOChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002105(CHEMBL192443)
Affinity DataKi:  0.870nMAssay Description:Binding affinity against Opioid receptor delta 1 from rat brain membranes using [3H]DADLEChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50404008(CHEMBL286693)
Affinity DataKi:  0.912nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Saint Louis University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50110941(1-(2,4-Dichloro-phenyl)-4-methyl-5-(4-pentyl-pheny...)
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]-CP-55,940 binding to cannabinoid receptor 1 in rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002116(CHEMBL363777)
Affinity DataKi:  1.10nMAssay Description:Binding affinity against Opioid receptor delta 1 from rat brain membranes using [3H]DADLEChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1136((4R,5R,6R)-6-benzyl-5-hydroxy-1-(1H-indazol-5-ylme...)
Affinity DataKi:  1.20nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
The State University Of New Jersey

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain membranes incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Saint Louis University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of [3H]-CP-55,940 binding to cannabinoid receptor 1 in rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM50473994(CHEMBL416964)
Affinity DataKi:  1.40nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
The State University Of New Jersey

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma-1 receptor in guinea pig brain membranes incubated for 1 hr in presence of 250 uM phenytoin liquid sc...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Missouri-St. Louis

Curated by ChEMBL
LigandPNGBDBM1093((4R,5R,6R)-Tetrahydro-1,3-bis[(4-fluoro-3-benzamid...)
Affinity DataKi:  1.40nMAssay Description:Inhibitory activity against HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Medicine & Dentistry Of New Jersey-Robert Wood Johnson Medical School (Umdnj-Rwjms)

Curated by ChEMBL
LigandPNGBDBM50002041(CHEMBL195784)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against Opioid receptor mu 1 from rat brain membranes using [3H]DAMGOChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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