TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.470nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.670nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Inhibition of rat TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.770nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.860nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.870nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Inhibition of arginylaminopeptidase (aminopeptidase B)More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.990nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 1nM ΔG°: -50.9kJ/molepH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
Affinity DataKi: 1nM ΔG°: -50.9kJ/molepH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2nM ΔG°: -49.2kJ/molepH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 3nM ΔG°: -48.2kJ/molepH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat kidney mitochondrial fractions incubated for 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 4nM ΔG°: -47.5kJ/molepH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Stanford University School Of Medicine
Curated by ChEMBL
Stanford University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
Affinity DataKi: 8nM ΔG°: -45.7kJ/molepH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of arginylaminopeptidase (aminopeptidase B)More data for this Ligand-Target Pair
Affinity DataKi: 12nM ΔG°: -44.8kJ/molepH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
Affinity DataKi: 30nM ΔG°: -42.5kJ/molepH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of p38alpha by spectrophotometric coupled enzyme assayMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibitory potency was measured on aminopeptidase N (APN)More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of aminopeptidase N (APN)More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Inhibitory potency was measured on aminopeptidase N (APN)More data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Inhibition of arginylaminopeptidase (aminopeptidase B)More data for this Ligand-Target Pair
Affinity DataKi: 56nM ΔG°: -41.0kJ/molepH: 7.5 T: 2°CAssay Description:The DPP activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 355 nm and meas...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of JNK3 by spectrophotometric coupled enzyme assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of JNK3 by spectrophotometric coupled enzyme assayMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibition of aminopeptidase N (APN)More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Inhibitory potency was measured on aminopeptidase N (APN)More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inihibitionof aminopeptidase A (APA)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
The University Of Mississippi
Curated by ChEMBL
The University Of Mississippi
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Displacement of [3H]mesulergine form human cloned 5HT2C receptor expressed in african green monkey COS7 cells by scintillation spectroscopyMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of aminopeptidase A (APA)More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inihibitionof aminopeptidase A (APA)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Inhibition of JNK3 by spectrophotometric coupled enzyme assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibition of JNK3 by spectrophotometric coupled enzyme assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 185nMAssay Description:Inhibition of JNK3 by spectrophotometric coupled enzyme assayMore data for this Ligand-Target Pair