TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.00560nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.00900nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0110nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0150nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0190nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0210nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0220nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0250nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0250nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0280nMAssay Description:Displacement of [125I]5-A-85380 from alpha4beta2 nicotinic receptor in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0280nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0310nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0310nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0340nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0350nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0350nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0350nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0410nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-6(Rattus norvegicus)
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0470nMAssay Description:Displacement of [3H]epibatidine from rat alpha6beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0500nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0580nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0610nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0610nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0620nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0620nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:In vitro affinity of the compound at the 5-HT reuptake site using [3H]-paroxetine as radioligand in rat frontal cortex membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0930nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0950nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-2(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.0950nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta4 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:In vitro affinity of the compound at the 5-HT reuptake site using [3H]-paroxetine as radioligand in rat frontal cortex membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]-Nal in rat brain homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine 1A receptor by [3H]-8-OH-DPAT displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Affinity at the 5-HT reuptake site labeled with [3H]-paroxetine using rat frontal cortex membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly
Curated by PDSP Ki Database
Eli Lilly
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Nida Addiction Research Center
Curated by PDSP Ki Database
Nida Addiction Research Center
Curated by PDSP Ki Database
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly
Curated by PDSP Ki Database
Eli Lilly
Curated by PDSP Ki Database
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]paroxetine from 5HT reuptake siteMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Affinity at the 5-HT reuptake site labeled with [3H]-paroxetine using rat frontal cortex membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity towards mu-opioid receptor by the displacement of [3H]-Nal in rat brain homogenatesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Rattus norvegicus (Rat))
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
The Johns Hopkins University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nicotinic receptor expressed in human HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair