Compile Data Set for Download or QSAR
maximum 50k data
Found 49 with Last Name = 'yang' and Initial = 'cn'
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50388392(CHEMBL2058262)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of GLUT1 mediated [3H]-2-DG uptake in human LNCAP cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50008923((S)-4-ethyl-4-hydroxy-1,12-dihydro-4H-2-oxa-6,12a-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326196((E)-6-Hydroxy-9-methoxy-11H-indeno[1,2-c]quinolin-...)
Affinity DataIC50:  3.76E+3nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50388391(CHEMBL2057965)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of GLUT1 mediated [3H]-2-DG uptake in human LNCAP cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326192((E)-9-methoxy-6-(piperazin-1-yl)-11H-indeno[1,2-c]...)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326187((E)-9-Methoxy-11H-indeno[1,2-c]quinolin-11-oneO-2-...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326181((E)-6-Hydroxy-9-methoxy-11H-indeno[1,2-c]quinolin-...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326186((E)-9-Methoxy-11H-indeno[1,2-c]quinolin-11-one O-2...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326191((E)-9-methoxy-6-(piperazin-1-yl)-11H-indeno[1,2-c]...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326194((E)-9-methoxy-6-(piperazin-1-yl)-11H-indeno[1,2-c]...)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326193((E)-9-methoxy-6-(piperazin-1-yl)-11H-indeno[1,2-c]...)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326195((E)-9-methoxy-6-(piperazin-1-yl)-11H-indeno[1,2-c]...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326184((E)-9-Methoxy-11H-indeno[1,2-c]quinolin-11-one O-2...)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM22984((8S,10S)-10-{[(2R,4S,5S,6S)-4-amino-5-hydroxy-6-me...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326185((E)-9-Methoxy-11H-indeno[1,2-c]quinolin-11-oneO-3-...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326182((E)-6-Hydroxy-9-methoxy-11H-indeno[1,2-c]quinolin-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326183((E)-9-Methoxy-11H-indeno[1,2-c]quinolin-11-oneO-2-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326189((E)-6-Hydroxy-9-methoxy-11H-indeno[1,2-c]quinolin-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326188(9-Methoxy-11H-indeno[1,2-c]quinolin-11-one | CHEMB...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50326190((E)-6-Hydroxy-9-methoxy-11H-indeno[1,2-c]quinolin-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human topoisomerase 1 assessed as decrease in pBR322 mobility on agarose gel by electrophoresisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPH domain leucine-rich repeat-containing protein phosphatase 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078209(CHEMBL3414686)
Affinity DataKd:  720nMAssay Description:Binding affinity to GST-tagged PH domain of PHLPP1 (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPH domain leucine-rich repeat-containing protein phosphatase 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078207(CHEMBL3414688)
Affinity DataKd:  690nMAssay Description:Binding affinity to GST-tagged PH domain of PHLPP1 (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078259(CHEMBL3414669)
Affinity DataKd:  1.02E+4nMAssay Description:Binding affinity to GST-tagged PH domain of PDK1 (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078209(CHEMBL3414686)
Affinity DataKd:  1.95E+4nMAssay Description:Binding affinity to GST-tagged PH domain of PDK1 (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078207(CHEMBL3414688)
Affinity DataKd:  1.11E+4nMAssay Description:Binding affinity to GST-tagged PH domain of PDK1 (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin-linked protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078259(CHEMBL3414669)
Affinity DataKd:  8.70E+3nMAssay Description:Binding affinity to GST-tagged PH domain of ILK (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin-linked protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078209(CHEMBL3414686)
Affinity DataKd:  6.20E+3nMAssay Description:Binding affinity to GST-tagged PH domain of ILK (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin-linked protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078207(CHEMBL3414688)
Affinity DataKd:  1.31E+4nMAssay Description:Binding affinity to GST-tagged PH domain of ILK (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPH domain leucine-rich repeat-containing protein phosphatase 1(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078259(CHEMBL3414669)
Affinity DataKd:  690nMAssay Description:Binding affinity to GST-tagged PH domain of PHLPP1 (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078259(CHEMBL3414669)
Affinity DataKd:  540nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078257(CHEMBL3414670)
Affinity DataKd:  520nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078256(CHEMBL3414671)
Affinity DataKd:  8.50E+3nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078223(CHEMBL3414672)
Affinity DataKd:  410nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078222(CHEMBL3414673)
Affinity DataKd:  350nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078221(CHEMBL3414674)
Affinity DataKd:  410nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078220(CHEMBL3414675)
Affinity DataKd:  320nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078219(CHEMBL3414676)
Affinity DataKd:  280nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078218(CHEMBL3414677)
Affinity DataKd:  450nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078217(CHEMBL3414678)
Affinity DataKd:  1.18E+3nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078216(CHEMBL3414679)
Affinity DataKd:  1.88E+3nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078215(CHEMBL3414680)
Affinity DataKd:  340nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078214(CHEMBL3414681)
Affinity DataKd:  390nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078213(CHEMBL3414682)
Affinity DataKd:  340nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078212(CHEMBL3414683)
Affinity DataKd:  980nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078211(CHEMBL3414684)
Affinity DataKd:  30nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078210(CHEMBL3414685)
Affinity DataKd:  210nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078209(CHEMBL3414686)
Affinity DataKd:  200nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078207(CHEMBL3414688)
Affinity DataKd:  220nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50078208(CHEMBL3414687)
Affinity DataKd:  350nMAssay Description:Binding affinity to GST-tagged PH domain of AKT (unknown origin) by surface Plasmon resonance spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed