TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 165nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 205nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 224nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 387nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 574nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 655nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.11E+3nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.45E+3nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.47E+3nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.73E+3nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 1.89E+3nMAssay Description:Alpha-2 adrenergic receptor binding affinity was tested against membrane preparations of rat brain using 0.2 nM [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Ohio State University
Curated by ChEMBL
Ohio State University
Curated by ChEMBL
Affinity DataKi: 9.22E+3nMAssay Description:Alpha-1 adrenergic receptor binding affinity in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+4nMAssay Description:Competitive inhibition of mushroom tyrosinase after 30 mins by Lineweaver-Burk double reciprocal plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Competitive inhibition of mushroom tyrosinase after 30 mins by Lineweaver-Burk double reciprocal plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.80E+4nMAssay Description:Competitive inhibition of mushroom tyrosinase after 30 mins by Lineweaver-Burk double reciprocal plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+4nMAssay Description:Competitive inhibition of mushroom tyrosinase after 30 mins by Lineweaver-Burk double reciprocal plot analysisMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of rat ASBT expressed in HEK293 cells assessed as inhibition of [3H]-taurocholate uptake after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of mouse ASBT expressed in HEK293 cells assessed as inhibition of [3H]-taurocholate uptake after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.302nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.302nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.302nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.302nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.372nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.447nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.490nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of mouse ASBT expressed in HEK293 cells assessed as inhibition of [3H]-taurocholate uptake after 90 mins by scintillation counting analysi...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.501nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.501nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.501nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.501nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.501nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Condition 2: Activated ERK2 activity was determined in an IMAP-FP assay (Molecular Devices). Using this assay format, the potency (IC50) of each comp...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.603nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.603nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.603nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.603nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.708nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.794nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.794nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Lanzhou University
Curated by ChEMBL
Lanzhou University
Curated by ChEMBL
Affinity DataIC50: 0.794nMAssay Description:Inhibition of human VEGFR2 after 60 minsMore data for this Ligand-Target Pair