Found 844 with Last Name = 'van westen' and Initial = 'gj' 
Affinity DataKi: 0.230nMAssay Description:Inhibition of mouse DAGL-alpha expressed in HEK293T cell membranes assessed as inhibition constant pre-incubated for 20 mins before PNP-butyrate subs...More data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Inhibition of mouse DAGL-alpha expressed in HEK293T cell membranes assessed as inhibition constant pre-incubated for 20 mins before PNP-butyrate subs...More data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Inhibition of mouse DAGL-alpha expressed in HEK293T cell membranes assessed as inhibition constant pre-incubated for 20 mins before PNP-butyrate subs...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 10nMAssay Description:Inhibition of mouse DAGL-alpha expressed in HEK293T cell membranes assessed as inhibition constant pre-incubated for 20 mins before PNP-butyrate subs...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]PSB-603 from human A2B receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]PSB-11 from human A3 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK 293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Ki values for sodium fluorescein (10 uM) uptake in OATP1B1-transfected CHO cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 61nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 69nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 71nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Ki values for sodium fluorescein (10 uM) uptake in OATP1B1-transfected CHO cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 83nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 105nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 106nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Displacement of [3H]-DPCPX from human A1 receptor expressed in CHO cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Ki values for sodium fluorescein (10 uM) uptake in OATP1B1-transfected CHO cellsMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Ki values for sodium fluorescein (10 uM) uptake in OATP1B3-transfected CHO cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 158nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 159nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK 293 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
Ku Leuven
Curated by ChEMBL
Ku Leuven
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Ki values for sodium fluorescein (10 uM) uptake in OATP1B1-transfected CHO cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 171nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 195nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 196nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Karlsruhe Institute Of Technology (Kit)
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in CHO-K1 cell membrane measured after 3 hrs by scintillation spectrometryMore data for this Ligand-Target Pair
