Affinity DataKi: 7.40nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes measured after 3 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity against human adenosine A2A receptor expressed in HEK293 cells using [3H]ZM-241385More data for this Ligand-Target Pair
Affinity DataEC50: 9.80nMAssay Description:Partial agonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as intrinsic activity by measuring cell index change withi...More data for this Ligand-Target Pair