Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetSialidase(Clostridium perfringens)
Graduate School Of Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50311743(CHEMBL487992 | GARTANIN)
Affinity DataKi:  3.60E+3nMAssay Description:Competitive inhibition of Clostridium perfringens neuraminidase by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase(Clostridium perfringens)
Graduate School Of Gyeongsang National University

Curated by ChEMBL
LigandPNGBDBM50311743(CHEMBL487992 | GARTANIN)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of Clostridium perfringens neuraminidase by fluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNEDD8-conjugating enzyme Ubc12(Homo sapiens)
Southwest Jiaotong University

Curated by ChEMBL
LigandPNGBDBM50311743(CHEMBL487992 | GARTANIN)
Affinity DataIC50:  1.03E+4nMAssay Description:Inhibition of Ubc12 (unknown origin)-neddylation incubated for 30 mins in presence of ATP by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTranscription factor p65(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50311743(CHEMBL487992 | GARTANIN)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of nuclear factor NF-kappa-B p65 subunit after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear factor NF-kappa-B p105 subunit(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50311743(CHEMBL487992 | GARTANIN)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of p50 after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed