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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetP2X purinoceptor 3(Homo sapiens (Human))
Beyer Aktiengesellschaft

US Patent
LigandPNGBDBM320251(3-(5-Ethyl-1,3- thiazol-2-yl)-5- {[(2S)-4- methylm...)
Affinity DataIC50:  23nMAssay Description:A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetP2X purinoceptor 2(Homo sapiens (Human))
Beyer Aktiengesellschaft

US Patent
LigandPNGBDBM320251(3-(5-Ethyl-1,3- thiazol-2-yl)-5- {[(2S)-4- methylm...)
Affinity DataIC50:  1.56E+3nMAssay Description:A fluorescent imaging plate reader (FLEX/FLIPR station; Molecular Devices) was used to monitor intracellular calcium levels using the calcium-chelati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent