Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1/2/3/4/5/6/7/8'
TargetMetabotropic glutamate receptor 1/2/3/4/5/6/7/8(Rattus norvegicus)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50132104(6-Methoxy-1-methyl-4,9-dihydro-3H-beta-carboline |...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1/2/3/4/5/6/7/8(Rattus norvegicus)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136493(1-Methyl-4,9-dihydro-3H-beta-carboline | 1-methyl-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1/2/3/4/5/6/7/8(Rattus norvegicus)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM100152(7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for rat 5-hydroxytryptamine 2A receptor using [3H]-DOBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1/2/3/4/5/6/7/8(Rattus norvegicus)
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50079183((2S)-amino(3,5-dihydroxyphenyl)ethanoic acid | (S)...)
Affinity DataEC50:  1.09E+4nMAssay Description:Compound was tested for ability to stimulate metabotropic glutamate receptor (mGluR) mediated phosphoinositide hydrolysis in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails