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Found 5 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 5 group A member 2' and Ligand = 'BDBM50605641'
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataKi:  0.150nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as inhibition con...More data for this Ligand-Target Pair
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TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataKd:  340nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataKd:  120nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataEC50:  43nMAssay Description:Agonist activity at LRH-1 (unknown origin) transfected in human HeLa cells measured after 24 hrs by Dual Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
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In DepthDetails PubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50605641(CHEMBL5177743)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to N-terminal 6-His tagged human LRH-1 LBD (299 to 541 residues) expressed in Escherichia coli BL21-(DE3) assessed as dissociation c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed