Affinity DataIC50: 2nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of rat NMDA receptor NR1C/NR2B subunit expressed in Xenopus laevis oocytes after 2 days by two-electrode voltage-clamp electrophysiologica...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Antagonistic activity against N-methyl-D-aspartate glutamate receptor 1/2B.More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Antagonist activity against rat 1A/2B subtype of N-methyl-D-aspartate(NMDA) receptor in xenopus oocytes.More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of rat NMDA receptor NR1F/NR2B subunit expressed in Xenopus laevis oocytes after 2 days by two-electrode voltage-clamp electrophysiologica...More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Antagonistic activity for suppression of membrane current response elicited by fixed concentration of glycine and glutamate in Xenopus oocyte express...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonist activity against rat 1A/2B subtype of N-methyl-D-aspartate(NMDA) receptor in xenopus oocytes.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of NMDA response at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Antagonistic activity for suppression of membrane current response elicited by fixed concentration of glycine and glutamate in Xenopus oocyte express...More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of NMDA response at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonistic activity for suppression of membrane current response elicited by fixed concentration of glycine and glutamate in Xenopus oocyte express...More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of NMDA response at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Antagonistic activity for suppression of membrane current response elicited by fixed concentration of glycine and glutamate in Xenopus oocyte express...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Functional antagonism by electrical assays in Xenopus oocytes expressing the 1A/2B NMDA receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of NMDA response at NR1A/2B receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity against rat 1A/2B subtype of N-methyl-D-aspartate(NMDA) receptor in xenopus oocytes.More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:In vitro inhibitory concentration against NMDA responses at NR1A/2B receptors expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Binding affinity against NR1A/2B receptor in rat brains by [3H]-ifenprodil displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Antagonist activity at wild type rat NR1/NR2B receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate/glycine-induced curren...More data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Antagonist activity at rat recombinant NR1/NR2B receptor expressed in frog oocytes assessed as inhibition of glutamate/glycine-induced current by two...More data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Antagonistic activity against N-methyl-D-aspartate glutamate receptor 1/2B.More data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibitory activity against Xenopus oocytes expressing rat N-Methyl-D-aspartate (NR1A/2B) Receptor subtype.More data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Compound was tested in vitro for inhibition of NMDA response at cloned NR1A/2A receptor expressed in Xenopus oocytesMore data for this Ligand-Target Pair