Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50312778
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50312778((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of rat GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash luminescence a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50312778((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50:  9.10nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50312778((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed