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Found 2 Enz. Inhib. hit(s) with Target = 'Growth hormone secretagogue receptor type 1' and Ligand = 'BDBM50312778'
TargetGrowth hormone secretagogue receptor type 1(Rattus norvegicus)
Amgen

Curated by ChEMBL
LigandPNGBDBM50312778((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of rat GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash luminescence a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50312778((S)-(4-(1H-indole-6-carbonyl)-3-methylpiperazin-1-...)
Affinity DataIC50:  9.10nMAssay Description:Antagonist activity at human GHSR expressed in CHOK1 cells assessed as inhibition of ghrelin-induced intracellular calcium flux by aequorin flash lum...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed