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Found 3 of ki for monomerid = 50387918
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM50387918(CHEMBL2058680 | US9283222, 459)
Affinity DataKi:  3nMpH: 8.0Assay Description:PARP1 assay was conducted in PARP assay buffer containing 50 mM Tris pH 8.0, 1 mM DTT, 4 mM MgCl2. PARP reactions contained 1.5 uM [3H]-NAD+ (1.6 uCi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM50387918(CHEMBL2058680 | US9283222, 459)
Affinity DataKi:  3nMAssay Description:Inhibition of PARP1 using [3H]NAD+ after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbvie

US Patent
LigandPNGBDBM50387918(CHEMBL2058680 | US9283222, 459)
Affinity DataKi:  3nMAssay Description:Binding affinity to PARP-1 (unknown origin) assessed as inhibition constant incubated for 1 hr by topcount microplate scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed