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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50056362'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50056362(3-Amino-5,6-dimethyl-2-[3-(4-pyrimidin-2-yl-pipera...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50056362(3-Amino-5,6-dimethyl-2-[3-(4-pyrimidin-2-yl-pipera...)
Affinity DataIC50:  6.80nMAssay Description:In vitro inhibitory concentration against radioligand [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor in rat hippocampal membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed