Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM34154'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universitat De Barcelona

LigandPNGBDBM34154(CHEMBL515307 | indenylsulfonamide, 15)
Affinity DataKi:  10nM ΔG°:  -47.5kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universitat De Barcelona

LigandPNGBDBM34154(CHEMBL515307 | indenylsulfonamide, 15)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universitat De Barcelona

LigandPNGBDBM34154(CHEMBL515307 | indenylsulfonamide, 15)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human 5HT6 receptor expressed in HEK293F cells assessed as stimulation of cAMP level after 30 mins by HTRF assay Inhibition of ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed