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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50266578'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50266578(CHEMBL477650 | N-{3-[2-(Dimethylamino)ethyl]-2-met...)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]LSD from human 5HT6 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Universitat De Barcelona

Curated by ChEMBL
LigandPNGBDBM50266578(CHEMBL477650 | N-{3-[2-(Dimethylamino)ethyl]-2-met...)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human 5HT6 receptor expressed in HEK293F cells assessed as stimulation of cAMP level after 30 mins by HTRF assay Inhibition of ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed