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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50300820'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50300820(CHEMBL565723 | N-(2-{3-[(3-Chlorophenyl)sulfonyl]-...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]LSD from human cloned 5HT6 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50300820(CHEMBL565723 | N-(2-{3-[(3-Chlorophenyl)sulfonyl]-...)
Affinity DataIC50:  8.30nMAssay Description:Antagonist activity at human cloned 5HT6 receptor expressed in HeLa cells assessed as inhibition of adenylyl cyclase activity by RIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed