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Found 16 Enz. Inhib. hit(s) with Target = '85/88 kDa calcium-independent phospholipase A2' and Ligand = 'BDBM50055366'
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  56nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free [14C]-AA formation after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  56nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free [14C]-AA formation after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  104nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  104nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in 16:0 LPC formation after 30 mins by HPLC-MS...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free AA formation after 30 mins by HPLC-MS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPC as substrate assessed as reduction in free AA formation after 30 mins by HPLC-MS ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPG as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPG as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPS as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  330nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPS as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as reduction in 16:0 LPC formation after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as assessed as reduction in free AA formation after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPE as substrate assessed as assessed as reduction in free AA formation after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPG as substrate assessed as reduction in free [14C]-AA formation after 30 mins in pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target85/88 kDa calcium-independent phospholipase A2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human recombinant calcium-independent PLA2 using PAPG as substrate assessed as reduction in free [14C]-AA formation after 30 mins in pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed