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Found 3 Enz. Inhib. hit(s) with Target = 'Acetylcholinesterase' and Ligand = 'BDBM50515460'
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad De Sevilla

Curated by ChEMBL
LigandPNGBDBM50515460(CHEMBL4475228)
Affinity DataKi:  75nMAssay Description:Inhibition of electric eel AChE assessed as dissociation constant for enzyme-inhibitor complex using acetylthiocholine iodide as substrate measured f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universidad De Sevilla

Curated by ChEMBL
LigandPNGBDBM50515460(CHEMBL4475228)
Affinity DataKi:  75nMAssay Description:Inhibition of electric eel AChE assessed as dissociation constant for enzyme-substrate-inhibitor complex using acetylthiocholine iodide as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universidad De Sevilla

Curated by ChEMBL
LigandPNGBDBM50515460(CHEMBL4475228)
Affinity DataIC50:  216nMAssay Description:Inhibition of human recombinant AChE expressed in HEK293 cells using acetylcholine iodide as substrate preincubated with enzyme for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed