Affinity DataKi: 9.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranes by competition association assayMore data for this Ligand-Target Pair
Affinity DataEC50: 7.60nMAssay Description:Agonist activity at human adenosine A1 receptor expressed in CHO cell membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair