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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50186599'
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50186599(8-cyclohexyl-2,6-diphenyl-9H-purine | CHEMBL207529...)
Affinity DataKi:  0.730nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50186599(8-cyclohexyl-2,6-diphenyl-9H-purine | CHEMBL207529...)
Affinity DataIC50:  477nMAssay Description:Activity against human adenosine A1 receptor in CHO cells assessed by the antagonizing effect of 100 nM CPA on forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed