Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50224760'
TargetAdenosine receptor A1(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50224760(2-chloro-N6-cyclopentyl-9H-(2-C-methyl-5-Nmethylca...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in pig cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
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Curated by ChEMBL
LigandPNGBDBM50224760(2-chloro-N6-cyclopentyl-9H-(2-C-methyl-5-Nmethylca...)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50224760(2-chloro-N6-cyclopentyl-9H-(2-C-methyl-5-Nmethylca...)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(GUINEA PIG)
Universit£

Curated by ChEMBL
LigandPNGBDBM50224760(2-chloro-N6-cyclopentyl-9H-(2-C-methyl-5-Nmethylca...)
Affinity DataEC50:  165nMAssay Description:Agonist activity at adenosine A1 receptor in pig cortical membrane assessed as stimulation of GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed