Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50267393'
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50267393(CHEMBL477444 | N6-Cyclopentyl-9H-(5-chloro-5-deoxy...)
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50267393(CHEMBL477444 | N6-Cyclopentyl-9H-(5-chloro-5-deoxy...)
Affinity DataKi:  0.720nMAssay Description:Binding affinity against Adenosine A1 receptor using [3H]CHA in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50267393(CHEMBL477444 | N6-Cyclopentyl-9H-(5-chloro-5-deoxy...)
Affinity DataKi:  9.5nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]DPCPX in rat cortical membranes in the absence of GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50267393(CHEMBL477444 | N6-Cyclopentyl-9H-(5-chloro-5-deoxy...)
Affinity DataKi:  62nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]DPCPX in rat cortical membranes in the presence of GTP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50267393(CHEMBL477444 | N6-Cyclopentyl-9H-(5-chloro-5-deoxy...)
Affinity DataEC50:  26nMAssay Description:Effective concentration for [35S]GTP-gamma-S, binding to adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed