Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a/A2b' and Ligand = 'BDBM50009702'
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50009702(2-Chloro-9-methyl-9H-purin-6-ylamine | CHEMBL31739...)
Affinity DataKi:  1.10E+4nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatum by using [3H]NECA as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50009702(2-Chloro-9-methyl-9H-purin-6-ylamine | CHEMBL31739...)
Affinity DataKi:  1.60E+4nMAssay Description:Tested for inhibition of rat PC12 adenylate cyclase stimulation by using NECA as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed