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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50059414'
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50059414(2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyri...)
Affinity DataKi: >100nMAssay Description:Binding affinity was determined in radioligand binding assay at rat striatal Adenosine A2A receptor vs [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50059414(2-Methyl-6-phenyl-4-phenylethynyl-1,4-dihydro-pyri...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity for adenosine A2A receptor as displacement of [3H]-CGS- 21680 from rat striatal membranes at 10e-4 MMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed