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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50078427'
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50078427(CHEMBL3414941)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]-NECA from human recombinant adenosine A2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50078427(CHEMBL3414941)
Affinity DataKi:  274nMAssay Description:Displacement of [3H]NECA from recombinant human adenosine A2A receptor expressed in CHO cell membranes after 3 hrs by microbeta scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50078427(CHEMBL3414941)
Affinity DataEC50:  22nMAssay Description:Agonist activity at recombinant human adenosine A2A receptor expressed in CHO cell membranes assessed as stimulation of adenylyl cyclase activity by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50078427(CHEMBL3414941)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human recombinant adenosine A2A receptor transfected in CHO cells assessed as induction of adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed