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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50187589'
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187589(CHEMBL3827859)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]MSX2 from adenosine receptor A2a in rat brain striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187589(CHEMBL3827859)
Affinity DataKi:  559nMAssay Description:Displacement of [3H]MSX2 from recombinant human adenosine receptor A2a expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50187589(CHEMBL3827859)
Affinity DataEC50:  460nMAssay Description:Antagonist activity at human adenosine receptor A2a expressed in CHO cell membranes assessed as inhibition of NECA-induced cAMP accumulation measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed