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Found 1 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50310912'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Vernalis (R&D)

Curated by ChEMBL
LigandPNGBDBM50310912((2-(pyridin-3-ylmethylamino)thieno[3,2-d]pyrimidin...)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at human adeosine A2A receptor expressed in CHOK1 cells assessed as inhibition of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed