Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM82032'
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataKi:  156nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataKi:  2.60E+3nMAssay Description:Binding affinity for adenosine A2A receptor from rat brain membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataKi:  2.70E+3nMAssay Description:Antagonism of cyclic [3H]AMP accumulation in guinea pig cerebral cortical slices (elicited by 15 uM 2-chloroadenosine at adenosine A2 receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataKi:  2.70E+3nMAssay Description:Compound was evaluated for its ability to antagonise cyclic [3H]-AMP accumulation in [3H]-adenine-labeled guinea pig cerebral cortical slices.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataKi:  3.00E+3nMAssay Description:Affinity against adenosine A2 receptor in the brain membranes measured by the displacement of [3H]-CPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataKi:  5.16E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University of Virginia

Curated by PDSP Ki Database
LigandPNGBDBM82032(1,3-Dipropyl-3,7-dihydro-purine-2,6-dione | 1,3-Di...)
Affinity DataEC50:  50nMAssay Description:Relexant activity on the spontaneous tone of isolated guinea pig tracheal ring chains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed