Affinity DataKi: 7.75nMAssay Description:Antagonist activity against human A2B adenosine receptor expressed in HEK-293 cells uisng [3H]-ZM-241,385 or [125I]-IABOPXMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity towards human Adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Displacement of [3H]DPCPX from human A2BAR expressed in HEK293 cell membrane incubated for 30 mins by microbeta trilux scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.41E+5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in human HEK293 cells incubated for 30 mins by fluorescence polarization bindin...More data for this Ligand-Target Pair