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Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50531422'
TargetAdenosine receptor A2b(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50531422(CHEMBL4522981)
Affinity DataIC50:  59nMAssay Description:Displacement of [3H]DPCPX from human A2B adenosine receptor expressed in HEK293 cell membranes after 60 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50531422(CHEMBL4522981)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at recombinant human A2B adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50531422(CHEMBL4522981)
Affinity DataIC50:  66nMAssay Description:Antagonist activity at human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A2b(Rattus norvegicus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50531422(CHEMBL4522981)
Affinity DataIC50:  280nMAssay Description:Antagonist activity at recombinant rat A2B adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Mus musculus)
Bayer Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50531422(CHEMBL4522981)
Affinity DataIC50:  400nMAssay Description:Antagonist activity at recombinant mouse A2B adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed