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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50170136'
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170136(1-Benzyl-7-ethyl-3-propyl-1H,6H-pyrrolo[2,1-f]puri...)
Affinity DataKi:  3.45nMAssay Description:Displacement of [3H]MRE3008F20 from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170136(1-Benzyl-7-ethyl-3-propyl-1H,6H-pyrrolo[2,1-f]puri...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170136(1-Benzyl-7-ethyl-3-propyl-1H,6H-pyrrolo[2,1-f]puri...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; range is 2.7 to 4.4 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170136(1-Benzyl-7-ethyl-3-propyl-1H,6H-pyrrolo[2,1-f]puri...)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as blockade of Cl-IB-MECA-mediated inhibition of forskolin-stimula...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed