Found 3 Enz. Inhib. hit(s) with Target = 'Aldo-keto reductase family 1 member C3' and Ligand = 'BDBM50337285'
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University of Pennsylvania
US Patent
University of Pennsylvania
US Patent
Affinity DataIC50: 120nMAssay Description:Compounds may be evaluated as selective reversible inhibitors of AKR1C3 by screening them against homogeneous recombinant AKR1C1-AKR1C4 expressed in ...More data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University of Pennsylvania
US Patent
University of Pennsylvania
US Patent
Affinity DataIC50: 120nMAssay Description:Inhibition of AKR1C3 by fluorimetric methodMore data for this Ligand-Target Pair
TargetAldo-keto reductase family 1 member C3(Homo sapiens (Human))
University of Pennsylvania
US Patent
University of Pennsylvania
US Patent
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant AKR1C3 assessed as NADP+ dependent oxidation of S-tetralol by fluorescence assayMore data for this Ligand-Target Pair