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Found 2 Enz. Inhib. hit(s) with Target = 'Aldo-keto reductase family 1 member C4' and Ligand = 'BDBM50382163'
TargetAldo-keto reductase family 1 member C4(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50382163(CHEMBL2023820)
Affinity DataIC50:  8.17E+3nMAssay Description:Inhibition of recombinant AKR1C4 assessed as enzyme catalyzed oxidation of S-tetralol by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member C4(Homo sapiens (Human))
Perelman School Of Medicine University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50382163(CHEMBL2023820)
Affinity DataIC50:  3.06E+4nMAssay Description:Inhibition of human AKR1C4 using S-tetralol as substrate in presence of NADP by fluorescence methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed