Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor' and Ligand = 'BDBM50019959'
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50019959(1-(4-Fluoro-phenyl)-4-[4-(2-methoxy-phenyl)-pipera...)
Affinity DataKi:  0.870nMAssay Description:Potency to displace [3H]- WB-4101 from alpha-1 adrenergic receptor in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50019959(1-(4-Fluoro-phenyl)-4-[4-(2-methoxy-phenyl)-pipera...)
Affinity DataKi:  0.870nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed