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Found 5 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50022722'
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataKi:  9.77E+3nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataKi:  9.77E+3nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataKi:  9.80E+3nMAssay Description:Binding affinity towards rat submaxillary gland Alpha-1 adrenergic receptor; value ranges from (6.2 - 15)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataEC50:  2.34E+5nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataEC50:  2.30E+5nMAssay Description:Effective concentration of the compound was determined in vitro against rabbit urethra Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed