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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-1D adrenergic receptor' and Ligand = 'BDBM50409813'
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50409813(CHEMBL1083181 | CHEMBL37883)
Affinity DataKi:  11nMAssay Description:Displacement of [3H] prazosin from human cloned adrenoceptor alpha 1D expressed in CHO cell membrane incubated for 30 mins by liquid scintillation co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50409813(CHEMBL1083181 | CHEMBL37883)
Affinity DataKi:  11.5nMAssay Description:Displacement of [3H]prazosin from human recombinant Alpha-1D adrenoreceptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50409813(CHEMBL1083181 | CHEMBL37883)
Affinity DataKi:  11.5nMAssay Description:Displacement of [3H]prazosin from human Alpha-1D adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed