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Found 4 Enz. Inhib. hit(s) with Target = 'Alpha-2B adrenergic receptor' and Ligand = 'BDBM50052880'
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataKi:  8.90nMAssay Description:Binding affinity for human Alpha-2B adrenergic receptor from cultured LM(tk-) cells using [3H]- prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Allergan

Curated by ChEMBL
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataKi:  17nMAssay Description:Compound was tested in vitro for binding affinity against Alpha-2B adrenergic receptor from cloned rat RNG receptor transfected into Chinese hamster ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Allergan

Curated by ChEMBL
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataKi:  17nMAssay Description:Displacement of rauwolscine from rat Alpha-2B adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50052880(CHEMBL49137 | Imidazolidin-2-ylidene-(5-methyl-qui...)
Affinity DataEC50:  78nMAssay Description:Alpha-2B adrenergic receptor agonistic potency as inhibition of forskolin-stimulated cyclic adenosine monophosphate synthesisMore data for this Ligand-Target Pair
In DepthDetails