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Found 2 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM50038942'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038942(CHEMBL63458 | N-(9,10,10-Trioxo-9,10-dihydro-10lam...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038942(CHEMBL63458 | N-(9,10,10-Trioxo-9,10-dihydro-10lam...)
Affinity DataIC50:  60nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]-5-HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed