Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM50038943'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))TBA
LigandPNGBDBM50038943(CHEMBL66260 | N-(7-Acetylamino-10-methyl-5,5-dioxo...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant MAO-AMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038943(CHEMBL66260 | N-(7-Acetylamino-10-methyl-5,5-dioxo...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]-5-HT at 1 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed