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Found 5 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] B' and Ligand = 'BDBM36551'
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
The Weizmann Institute of Science

LigandPNGBDBM36551(Chelator, M30 | US9034303, M30)
Affinity DataIC50:  37nMpH: 7.4 T: 2°CAssay Description:Inhibition of MAO activity in rat brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM36551(Chelator, M30 | US9034303, M30)
Affinity DataIC50:  57nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
The Weizmann Institute of Science

LigandPNGBDBM36551(Chelator, M30 | US9034303, M30)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of MAO-B in rat liver homogenate using [14C]-phenylethylamine as substrate preincubated for 30 mins followed by substrate addition measure...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM36551(Chelator, M30 | US9034303, M30)
Affinity DataIC50:  1.50E+3nMAssay Description:Mixed type inhibition of MAOB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM36551(Chelator, M30 | US9034303, M30)
Affinity DataIC50:  1.02E+4nMAssay Description:Irreversible inhibition of MAOB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed