Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM18545'
TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

LigandPNGBDBM18545(7-[(2-methylpropyl)amino]-4-(trifluoromethyl)-1,2-...)
Affinity DataKi:  65nM ΔG°:  -42.7kJ/mole IC50:  74nMpH: 7.4 T: 2°CAssay Description:The compounds were evaluated in a transcriptional activation assay with hAR in a mammalian cell background (CV-1) as the primary in vitro assay. Rece...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed