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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50204245'
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50204245(CHEMBL3898284)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]DHT from androgen receptor in human MDA-MB-453 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50204245(CHEMBL3898284)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of testosterone-induced transactivationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed