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Found 2 Enz. Inhib. hit(s) with Target = 'Androgen receptor' and Ligand = 'BDBM50430944'
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430944(CHEMBL2336966)
Affinity DataIC50:  1.46E+3nMAssay Description:Displacement of [3H] ]5alpha-DHT from mouse androgen receptor expressed in monkey COS7 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Mus musculus)
Chonnam National University

Curated by ChEMBL
LigandPNGBDBM50430944(CHEMBL2336966)
Affinity DataIC50:  4.45E+3nMAssay Description:Agonist activity at mouse androgen receptor assessed as inhibition of transactivation after 24 hrs by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed