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Found 2 Enz. Inhib. hit(s) with Target = 'Apelin receptor' and Ligand = 'BDBM50571395'
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50571395(CHEMBL4862328)
Affinity DataEC50:  3.40E+3nMAssay Description:Agonist activity at human AGTRL1 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50571395(CHEMBL4862328)
Affinity DataEC50:  241nMAssay Description:Agonist activity at human APJ receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 40 mins by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed